DMPK(药物代谢和药代动力学)

DMPK(药物代谢和药代动力学)分析是药物研发阶段的重要组成部分:从数个成药的候选对象中选择生物利用度最高,生物安全性最好,治疗效果最佳的对象,DMPK实验的成败将决定的在研候选药物是否能够在通向市场的路上走下去,而DMPK实验室数据的安全有效的管理正面临着挑战! 

如何能够合理设计与某个研究对象相关的所有研究和测试,并根据实验人员的不同身份进行工作的安排?如何能够保证DMPK实验室数据的安全管理,数据不会被随意改动?如何能够保证对样品的管理准确有效?如何能够让负责DMPK工作的CRO企业与制药公司互相沟通?如何保证DMPK工作的数据信息能够通过严格FDA审核,提高制药公司DMPK的研究效率,增加CRO企业的国际竞争能力? 

我现在只需要是利用是码把蛋白质中的分子欧几里得距离计算出来,输出结果是一个二维的矩阵 现在缺少一个数据集 只有一个p: site AAK1: [74,176] ABL1(E255K): [308] ABL1(F317I): [308] ABL1(F317I)p: [308] ABL1(F317L): [308] ABL1(F317L)p: [308] ABL1(H396P): [308] ABL1(H396P)p: [308] ABL1(M351T): [308] ABL1(Q252H): [308] ABL1(Q252H)p: [308] ABL1(T315I): [308] ABL1(T315I)p: [308] ABL1(Y253F): [308] ABL1: [308] ABL1p: [308] ABL2: [302] ACVR1: [235,336] ACVR1B: [234,335] ACVR2A: [219,322] ACVR2B: [217,321] ACVRL1: [229,330] ADCK3: [340,358,488,493,507] ADCK4: [219,237,367,372,386] AKT1: [53,86,179,234,278,292] AKT2: [188] AKT3: [187] ALK: [1124,1150,1199] AMPK-alpha1: [56,150] AMPK-alpha2: [45,139] ANKK1: [51,145] ARK5: [84,178] ASK1: [709,803] ASK2: [677,771] AURKA: [143,162,256,274] AURKB: [106,200] AURKC: [72,166] AXL: [567,672] BIKE: [79,180] BLK: [269] BMPR1A: [261,362] BMPR1B: [231,332] BMPR2: [230,333,351] BMX: [445,536] BRAF: [483,576] BRAF(V600E): [483,576] BRK: [219,312] BRSK1: [63,156] BRSK2: [48,141] BTK: [26,28,39,53,430] CAMK1: [49,141] CAMK1D: [52,144] CAMK1G: [52,143] CAMK2A: [42,135] CAMK2B: [43,136] CAMK2D: [43,136] CAMK2G: [43,136] CAMK4: [75,164] CAMKK1: [157,275] CAMKK2: [194,312] CASK: [41,141] CDC2L1: (563) CDC2L2: (261) CDC2L5: (208) CDK11: [52,151] CDK2: [33,86,127,145] CDK3: [33,127] CDK4-cyclinD1: [35,140] CDK4-cyclinD3: [35,140] CDK5: [33,126] CDK7: [41,137] CDK8: [52,151] CDK9: [48,149,167] CDKL1: [34] CDKL2: [33,126] CDKL3: [33,125] CDKL5: [43] CHEK1: [38,130] CHEK2: [249,347,368] CIT: [126,221] CLK1: [191,288] CLK2: [193,290] CLK3: [334,431] CLK4: [189,286] CSF1R: [616,778] CSK: [222,314] CSNK1A1: [46,136] CSNK1A1L: [46,136] CSNK1D: [38,128] CSNK1E: [38,128] CSNK1G1: [73,164] CSNK1G2: [75,165] CSNK1G3: [72,117,119,162] CSNK2A1: [68,156] CSNK2A2: [69,157] CTK: [262,352] DAPK1: [42,100,139,161] DAPK2: [52,149] DAPK3: [42,94,96,139] DCAMKL1: [419,511] DCAMKL2: [423,515] DCAMKL3: [385,477] DDR1: [655,766] DDR2: [608,710] DLK: [152,236] DMPK: [100,195] DMPK2: [100,195] DRAK1: [90,186] DRAK2: [62,158] 我现在应该怎么办?
最新发布
03-25
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